Selected Publications: |
- “Click” ligand for “Click” chemistry: (1-(4-Methoxybenzyl)-1-H-1, 2, 3-triazol-4-yl) methanol (MBHTM) accelerated Copper-catalyzed [3+2] Azide-Alkyne cycloaddition (CuAAC) at low catalyst loading. Rajesh H. Tale, Venkatesh B. Gopula , Gopal K. Toradmal. Tetrahedron Lett. 2015, 56, 5864–5869 IF 2.39
- A Practical and General Ipso Iodination of Arylboronic Acids Using N–Iodomorpholinium Iodide (NIMI) as a Novel Iodinating Agent: Mild and Regioselective Synthesis of Aryliodides. H. Tale, G. K. Toradmal, V. B. Gopula. RSC Advances, 2015, 5, 84910-84919 IF 3.85
- Metal free Ipso Iodination of Arylboronic Acids Using CTAB / I2 In Aqueous Media: Green and Regioselective Synthesis of Aryl iodides Under Mild Conditions. Rajesh Tale, Gopal Toradmal, Venkatesh Gopula, Atish H. Rodge, Rajendra P. Pawar , Kalpana M. Patil , Tetrahedron Lett. 2015, 56, 2699–2703, IF= 2.379
- Synthesis and Biological Evaluation of Novel 2’,4’,5’-Trimethoxyflavonal Derivatives as Anti-inflammatory and Antimicrobial Agents. Hantapure, G. D., Keche, A. P., Rodge, A. H., Tale, R. H., Birajdar, S. S., Pawar, M.J., Kamble, V. M. Medicinal Chemistry Resrach, 2013. IF 1.4
- A Novel Pyrazole Derivatives with Aryl Urea, Thiourea and Sulfonamide Moieties: Synthesis, Anti-inflammatoty and Antimicrobial Evaluation. Ashish P. Keche, Girish D. Hantapure, Rajesh H. Tale, Atish H. Rodge, Satish S. Biragar, Vandana M. Kamble. Biorganic & Medicinal Chemistry Letter, 2012, 22, 6611-6615 IF 2.42
- Synthesis and Biological Evaluation of Novel Piperazine Derivatives of Flavones as Potent Anti-inflammatory and Antimicrobial Agents. Rajesh H. Tale, Ashish P. Keche, Girish D. Hantapure, Atish H. Rodge, Vandana M. Kamble. Biorganic & Medicinal Chemistry Letter, 2012,22, 6385-6390 IF 2.42
- Synthesis, Anti-inflammatory and Antibacterial Evaluation of Novel N1-(Quinolin-4-yl)ethane-1,2-diamine Phenyl Urea derivatives. Keche A. P., Hantapure, G. D. Tale R. H., Rodge A. H. Chem. Res. 2012, 22(3),1480-1487 IF 1.4
- A Novel pyrimidine derivatives with aryl urea, thiourea and sulfonamide moieties: Synthesis , anti-inflammatoty and antimicrobial evaluation. Ashish P. Keche, Girish D. Hantapure, Rajesh H. Tale, Atish H. Rodge, Satish S. Biragar, Vandana M. Kamble. Biorganic & Medicinal Chemistry Letter, 2012, 22, 3445-3448 IF 2.42
- The synthesis, anti-inflammatory, and anti-microbial activity evaluation of new series of 4-(3-arylureido)phenyl-1,4-dihydropyridine derivatives. Rajesh H. Tale, Atish H. Rodge, Girish D. Hantapure, Ashish P. Keche, Kalpana, M. Patil, Rajendra P. Pawar. Chem. Res. 2013, 22 (3), 1450-1455
- IF 1.4
- The synthesis, anti-inflammatory and antimicrobial activity evaluation of novel thioanalogues of 3, 4-dihydropyrimidin-2(1-H)-one urea derivatives of N-aryl ureas. Rajesh H. Tale, Atish H. Rodge, Girish D. Hantapure, Ashish P. Keche, Kalpana, M. Patil, Rajendra P. Pawar. Chem. Res. 2012,21,4152-4260
- IF 1.4
- A robust, simple and rapid validated method for estimation of erythromycin ethylsuccinate in human plasma by liquid chromatography - tandem mass spectrometry and its application to clinical study. Arvind G. Jangid, Rajesh H. Tale , Vikas V. Vaidya. International of Pharmaceutical pharmulations and Analysis. 2011, 2, 1-7
- The Novel 3, 4-Dihydropyrimidin-2(1-H)-one urea derivatives of N-aryl urea: Synthesis, anti-inflammatory, antibacterial and antifungal activity evaluation. Rajesh H. Tale, Atish H. Rodge, Girish D. Hatnapure, Ashish P. Ketches, Bioorganic and Medicinal Chemistry Letters (BMCL) 2011,21, 4648-4651.
- IF 2.42
- Single, Selective and Simple Validated Method for Simultanious Estimation of Amiloride and Hydrochorothiaziden in Human Plasma by Liquid Chromatography-Tendem Mass Spectrometry. Rajesh H. Tale, Vikas. V. Vaidya and Arvind G. Jangid. Biomedical Chromatography. 2012, 26, 95-100. IF 1.79
- Estimation of Two Bioactive Compounds From Artocarpus Lakoocha Roxb. Leaves Using HPTLC. Ashish Raote, Arivnd Jangid, Rajesh Tale, International Journal of Pharma and Bio Sciences 2011, 2, 861-866.
- Liquid Chromatography-Tandem Mass Spectrometric Method For Simultaneous Determination of Rutin and Qercetin From Leaves of Artocarpus Lakoocha Ashish Raote, Arvind Jangid, Rajesh Tale, Vikas. V. Vaidya. International Journal of Pharma and Bio Sciences 2011, 2, 848-853.
- Synthesis and evaluation of anti-bacterial, anti-fungal activities of novel, 2, 4-Oxadiazoles. Rajesh H. Tale, Atish H. Rodge, Girish D. Hatnapure, Ashish P. Keche, Pramod R. Padole. Chem. Pharm. Res., 2011, 3(2): 496-505
- A simple, selective and rapid validated method for estimation of anastrazole in human plasma by liquid chromatography-tendem mass spectrometry and its application to bioequivalence study. Arvind G Jangid, Ashutosh M. Pudge , Santosh, S. Joshi , Pramod N. Pabrekar, Rajesh H. Tale and Vikas V. Vaidya. Biomedical Chromatography. 2010, 24, 727-731. IF 1.79
- A novel 3-nitrobenzeneboronic acid as an extremely mild and environmentally benign catalyst for the acetylation of alcohols under solvent-free conditions.Tale, R.H., Adude, R.N. Tetrahedron Letters ,2006, 47 , 7263-7265. IF 2.379
- 3-Nitrobenzeneboronic acid as an efficient and environmentally benign catalyst for the selective transesterification of β-keto esters. Tale, R.H., Sagar, A.D., Santan, H.D., Adude, R.N., Synlett, 2006, (3). 415-418. IF 2.379
- Synthesis of symmetrical diaryl ethers from arylboronic acids mediated by copper(II) acetate Sagar, A.D., Tale, R.H., Adude, R.N. , Tetrahedron Letters, 2003, 44, 7061-7063. IF 2.379
- An extremely simple, convenient and mild one-pot reduction of carboxylic acids to alcohols using 3,4,5-trifluorophenylboronic acid and sodium borohydride.Tale, R.H., Patil, K.M., Dapurkar, S.E., Tetrahedron Letters, 2003, 44, 3427-3428. IF 2.379
- 3,4,5-Trifluorobenzeneboronic acid: A mild and versatile catalyst for the one-pot synthesis of acyl azides from carboxylic acids Tale, R.H., Patil, K.M. Tetrahedron Letters,2002, 43, 9715-9716. IF 2.379
Book Chapter published
Published a chapter on boronic acids (3-Nitrophenylboronic acid) in the “ Electronic Encyclopedia of Regents in Organic Synthesis (e-EROS)” published by John-Wiley-Interscience in 2009.( Honorium $ 150).
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